A novel acetylated analogue of dynorphin A-(1-11) amide as a kappa-opioid receptor antagonist

J Med Chem. 1999 Aug 12;42(16):3011-3. doi: 10.1021/jm9901071.
No abstract available

Publication types

  • Letter
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • CHO Cells
  • Cricetinae
  • Dynorphins / chemistry*
  • Oligopeptides / chemical synthesis*
  • Oligopeptides / chemistry
  • Oligopeptides / pharmacology
  • Peptide Fragments / chemistry*
  • Radioligand Assay
  • Receptors, Opioid, kappa / antagonists & inhibitors*

Substances

  • Oligopeptides
  • Peptide Fragments
  • Receptors, Opioid, kappa
  • dynorphin A (1-11)-amide
  • JVA 901
  • Dynorphins